BiKin 1

BiKin 1 is a new kinase inhibitor Library (1000cpds).  It’s based on a new scaffold which allow high chemical diversity and high-throughput synthesis. The activity (% inhibition at 10uM) of 18 cpds has been evaluated in a panel of 50 kinases.

—On 815 generated data points at 10uM:

—45 points with a % Inh>20%

—21 with a % Inh>30%

—10 with a % Inh>50%

—Best is 84% inh at 10uM.

These data confirm the great potential of the Bikin 1 library.

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