BiKin 1 is a new kinase inhibitor Library (1000cpds). It’s based on a new scaffold which allow high chemical diversity and high-throughput synthesis. The activity (% inhibition at 10uM) of 18 cpds has been evaluated in a panel of 50 kinases.
On 815 generated data points at 10uM:
45 points with a % Inh>20%
21 with a % Inh>30%
10 with a % Inh>50%
Best is 84% inh at 10uM.
These data confirm the great potential of the Bikin 1 library.
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